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CAS No.: 483-14-7
Synonyms: (-)-Tetrahydropalmatine;L-Tetrahydropalmatine;(–)-Corydalis B
Rotundine is antagonist for domapmine D1 receptor(Ki = 124 nM) and has a lower binding activity of domapmine D2 receptor and domapmine D3 receptor. It can also inhibit 5-HT1A (Ki = 340 nM).
规格 | 价格 | 促销价格 | 库存 | 数量 |
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01631383 | Cocaine Use | Phase 1 | Completed | - | United States, Maryland ... more >> Maryland Psychiatric Research Center Catonsville, Maryland, United States, 21228 Collapse << |
NCT02118610 | Schizophrenia | Not Applicable | Recruiting | December 2019 | United States, Maryland ... more >> Maryland Psyciatric Research Center Recruiting Catonsville, Maryland, United States, 21228 Contact: Ann Kearns, BS 410-402-6854 akearns@mprc.umaryland.edu Collapse << |
NCT02139761 | Cocaine Use | Phase 2 | Withdrawn(Study funding has no... more >>t been established) Collapse << | June 2016 | United States, Maryland ... more >> Maryland Psychiatric Research Center Catonsville, Maryland, United States, 21228 Collapse << |
实验方案
技术信息
CAS号 | 483-14-7 | 储存条件 |
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分子式 | C21H25NO4 | 运输 | 蓝冰 | |||||
分子量 | 355.43 | 别名 | (-)-Tetrahydropalmatine;L-Tetrahydropalmatine;(–)-Corydalis B;(–)-Tetrahydropalmatine;(S)-Tetrahydropalmatine;L-THP;罗通定;延胡索乙素 | |||||
溶解度 |
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动物实验配方 |